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Showing 1-20 of 20 results for "476994" within Papers
A practical large-scale preparation of 5'-bromospiro (cyclohexane-1,3-[3H] indol)-2'(1'H)-one.
Wilk BK, et al.
Organic preparations and procedures international, 37(3), 283-285 (2005)
A green approach for efficient synthesis of N-substituted pyrroles in ionic liquid under microwave irradiation.
Meshram HM, et al.
Tetrahedron Letters, 51(27), 3477-3480 (2010)
Razieh Sabet et al.
European journal of medicinal chemistry, 45(3), 1113-1118 (2010-01-09)
Quantitative structure activity relationships (QSAR) of anti-cancer isatin derivatives were discovered by multiple linear regressions (MLR) and genetic algorithm partial least squares (GA-PLS) methods. Topological, chemical, geometrical and functional groups descriptors were found to be effective parameters on the cytotoxic
Synthesis of isatin and 5-bromoisatin derivatives.
Mesropyan EG, et al.
Russ. J. Org. Chem., 37(10), 1476-1477 (2001)
David Rudd et al.
Scientific reports, 5, 13408-13408 (2015-09-02)
Despite significant advances in chemical ecology, the biodistribution, temporal changes and ecological function of most marine secondary metabolites remain unknown. One such example is the association between choline esters and Tyrian purple precursors in muricid molluscs. Mass spectrometry imaging (MSI)
Synthesis, characterization and cytotoxic activity of S-benzyldithiocarbazate Schiff bases derived from 5-fluoroisatin, 5-chloroisatin, 5-bromoisatin and their crystal structures.
Manan MAFA, et al.
Journal of Chemical Crystallography, 41(11), 1630-1641 (2011)
Possible psychopharmacological agents. X. Synthesis of Some Fluorine Containing Indole-2, 3-dione Derivatives.
Joshi KC, et al.
J. Prakt. Chem., 322(2), 314-320 (1980)
V N Garalene et al.
Voprosy meditsinskoi khimii, 30(5), 56-59 (1984-09-01)
Effect of isatin and of three its derivatives on content of lactate, pyruvate and glycogen was studied in rat tissues. The substances studied, except of 5-butylisatin, decreased the content of lactic acid with simultaneous increase of glycogen content in liver
A facile one-pot method for the preparation of N-alkyl isatins under microwave irradiation.
Azizian J, et al.
Synthetic Communications, 33(5), 789-793 (2003)
SiO2 mediated reaction of isatin with N-halosaccharins: A regiospecific preparation of 5-haloisatins.
de Souza SPL, et al.
Heterocyclic Communications, 9(1), 31-34 (2003)
Superelectrophiles in aromatic polymer chemistry.
Colquhoun HM, et al.
Macromolecules, 34(4), 1122-1124 (2001)
Electro-organic synthesis of nanosized particles of 3-hydroxy-3-(1H-indol-3-yl) indolin-2-one derivatives.
Makarem S, et al.
Monatshefte fur Chemie / Chemical Monthly, 148(8), 1157-1160 (2012)
Cornelius Klöck et al.
Bioorganic & medicinal chemistry letters, 21(9), 2692-2696 (2011-01-11)
Inhibitors of human transglutaminase 2 (TG2) are anticipated to be useful in the therapy of a variety of diseases including celiac sprue as well as certain CNS disorders and cancers. A class of 3-acylidene-2-oxoindoles was identified as potent reversible inhibitors
Janice L Hyatt et al.
Journal of medicinal chemistry, 50(8), 1876-1885 (2007-03-24)
Carboxylesterases (CE) are ubiquitous enzymes thought to be responsible for the metabolism and detoxification of xenobiotics. Numerous clinically used drugs including Demerol, lidocaine, capecitabine, and CPT-11 are hydrolyzed by these enzymes. Hence, the identification and application of selective CE inhibitors
Synthesis and spectral data for cinchoninic acids.
Sarkis GY.
Journal of Chemical and Engineering Data, 17(3), 388-391 (1972)
Cale C Streeter et al.
Biochemistry, 58(17), 2260-2268 (2019-04-10)
The continued rise of antibiotic-resistant infections coupled with the limited pipeline of new antimicrobials highlights the pressing need for the development of new antibacterial agents. One potential pathway for new agents is de novo purine biosynthesis as studies have shown
Kara L Vine et al.
Bioorganic & medicinal chemistry, 15(2), 931-938 (2006-11-08)
A range of substituted 1H-indole-2,3-diones (isatins) were synthesized using standard procedures and their cytotoxicity evaluated against the human monocyte-like histiocytic lymphoma (U937) cell line in vitro. SAR studies identified C(5), C(6), and C(7) substitution greatly enhanced activity with some di-
The Structures of the Bromodioxindoles of Baeyer and Knop.
Sumpter WC.
Journal of the American Chemical Society, 67(7), 1140-1141 (1945)
V Garalene
Eksperimental'naia i klinicheskaia farmakologiia, 62(3), 20-24 (1999-08-10)
The inotropic activity of 5-bromisatin (5-bromindolyn-2,3-dion) which possesses antihypoxic properties was studied on rhythmically stimulated papillary muscles of guinea pigs, and the changes in the force of their contractions were recorded. The inotropic efficacy (calculated according to ED50 value) of
Quick and efficient synthesis of Morita-Baylis-Hillman adducts of isatin derivatives.
Rad-Moghadam K and Youseftabar-Miri L.
ARKIVOC (Gainesville, FL, United States), 11, 43-50 (2011)
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