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Merck
모든 사진(1)

문서

A6226

Sigma-Aldrich

AM251

>98% (HPLC), solid, cannabinoid receptor (CB1) antagonist

동의어(들):

1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide

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모든 사진(1)

About This Item

실험식(Hill 표기법):
C22H21N4OCl2I
CAS Number:
183232-66-8
Molecular Weight:
555.24
MDL number:
MFCD01861181
UNSPSC 코드:
12352200
PubChem Substance ID:
24891069
NACRES:
NA.77

product name

AM251, >98% (HPLC), solid

Quality Level

100

분석

>98% (HPLC)

형태

solid

색상

white

solubility

DMSO: >10 mg/mL
H2O: insoluble

주관자

Sanofi Aventis

SMILES string

Cc1c(nn(-c2ccc(Cl)cc2Cl)c1-c3ccc(I)cc3)C(=O)NN4CCCCC4

InChI

1S/C22H21Cl2IN4O/c1-14-20(22(30)27-28-11-3-2-4-12-28)26-29(19-10-7-16(23)13-18(19)24)21(14)15-5-8-17(25)9-6-15/h5-10,13H,2-4,11-12H2,1H3,(H,27,30)

InChI key

BUZAJRPLUGXRAB-UHFFFAOYSA-N

유전자 정보

mouse ... Cnr1(12801) , Cnr2(12802)
rat ... Cnr1(25248)

애플리케이션

AM251, a CB1 cannabinoid receptor antagonist, has been used in a study to determine its interaction with hippocampal neurons to enhance spatial memory in mice.

생화학적/생리학적 작용

AM251 is a CB1 cannabinoid receptor antagonist.

특징 및 장점

This compound is featured on the Cannabinoid Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
This compound was developed by Sanofi Aventis. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

기타 정보

Salt content may vary.

유해 및 위험 성명서

H413

예방조치 성명서

P273 - P501

Hazard Classifications

Aquatic Chronic 4

Storage Class Code

11 - Combustible Solids

WGK

WGK 3

Flash Point (°F)

Not applicable

Flash Point (°C)

Not applicable

개인 보호 장비

dust mask type N95 (US), Eyeshields, Gloves

시험 성적서(COA)

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이미 열람한 고객

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Sigma-Aldrich

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Sigma-Aldrich

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