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Merck
모든 사진(1)

주요 문서

SMB00947

Sigma-Aldrich

N-Desethyl amodiaquine dihydrochloride

≥95%

동의어(들):

Monodesethylamodiaquine dihydrochloride

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About This Item

실험식(Hill 표기법):
C18H18ClN3O · 2HCl
CAS Number:
Molecular Weight:
400.73
UNSPSC 코드:
41116107
NACRES:
NA.77

생물학적 소스

synthetic

Quality Level

분석

≥95%

양식

solid

분자량

400.73 g/mol

기술

HPLC: suitable

색상

yellow to dark yellow

solubility

DMSO: soluble
methanol: soluble
water: soluble

저장 온도

2-8°C

애플리케이션

Amodiaquine (AQ) is currently used in combination with Artesunate (AS) as first-line treatment for some cases of falciparum malaria (UM) in many countries. AQ is metabolized by hepatic cytochrome P450 2C8 (CYP2C8) to Desethylamodiaquine (DAQ; DEAQ; NADQ; Ndes-amo), which is subsequently eliminated via extra-hepatic biotransformation by CYP1A1 and CYP1B1. DEAQ is responsible for the pharmacological activity of AQ (both therapeutic and toxicity) due to its long elimination half-life.
Metabolomics research

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Storage Class Code

11 - Combustible Solids

WGK

WGK 3

Flash Point (°F)

Not applicable

Flash Point (°C)

Not applicable


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문서 라이브러리 방문

Yangshun Tang et al.
Toxicology in vitro : an international journal published in association with BIBRA, 62, 104669-104669 (2019-10-20)
Amodiaquine (ADQ), an antimalarial drug used in endemic areas, has been reported to be associated with liver toxicity; however, the mechanism underlying its hepatoxicity remains unclear. In this study, we examined the cytotoxicity of ADQ and its major metabolite N-desethylamodiaquine
Ahmed A Albassam et al.
Saudi pharmaceutical journal : SPJ : the official publication of the Saudi Pharmaceutical Society, 27(3), 406-412 (2019-04-13)
Pterostilbene is a natural polyphenol compound found in small berries that is related to resveratrol, but has better bioavailability and a longer half-life. The purpose of this study was to assess the potential inhibitory effect of pterostilbene on in vitro
Yingshan Han et al.
Journal of medical virology, 91(7), 1182-1190 (2019-02-26)
Studies aimed at repurposing existing drugs revealed that some antimalarial compounds possess anti-Zika virus (anti-ZIKV) activity. Here, we further tested 14 additional antimalarial drugs and their metabolites or analogs for anti-ZIKV activity using a phenotypic screening approach. We identified four

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